Ibisobanuro:
Urapidil hydrochloride ni umunwa ukora α1-adrenoeptor antagonist na 5-HT1A reseptor agonist hamwe na pIC50 ya 6.13 na 4.38 kurwanya α1- na α2-adrenoeptor. Urapidil hydrochloride yerekana ingaruka zidasanzwe.
Kunxiangda agaragara nk'umuyobozi ukomeye muri urwo rwego nk'umuntu utanga Urapidil hydrochloride, ibikomoka ku miti ikomeye. Azwi cyane kubera kwiyemeza ubuziranenge, Kunxiangda yishimiye afite icyemezo cya GMP, gihamya ko yubahiriza uburyo bukomeye bwo gukora ibicuruzwa. Iki cyemezo cyahawe isosiyete n’icyubahiro CFDA (Ubushinwa bushinzwe ibiryo n’ibiyobyabwenge mu Bushinwa), gishimangira ubwitange bwa Kunxiangda mu gukomeza amahame yo mu rwego rwo hejuru mu bicuruzwa no kubungabunga umutekano n’ibicuruzwa byabo.
Synonyme yicyongereza: 6 [[3- 6 - [[3- [4- (2-METHOXYPHENYL) -1-PIPERAZINYL] PROPYL] AMINO] -1,3-DIMETHYL-2,4 (1H, 3H) -PYRIMIDINEDIONE; 6 - [[3- [4- (2-METHOXYPHENYL) -1-PIPERAZINYL] PROPYL] AMINO] -1,3-DIMETHYL-2, 4 (1H, 3H) -PYRIMIDINEDIONEHYDROCHLORIDE; URAPIChemicalbookDILHCL; URAPIDILHYDROCHLORIDE; URAPIDILHYDROCHLORIDEA1ADRENOCEPTORANTAG; 6- [3- [4- (2-mikorerexyphenyl) piperazin-1-yl] propylamino] -1,3-dimethyl-pyrimidine-2,4-dionehydrochloride; 6- [3- [4- (2-mikorerexyphenyl) piperazin-1-yl] propylamino] -1,3-dimethylpyrimidine-2,4-dionehydrochloride
Amakuru ya tekiniki
CAS No: 64887-14-5
Inzira ya molekulari: c20h30cln5o3
Uburemere bwa molekuline: 423.94
EINECS No.: 636-348-0
Kugaragara: Birakomeye
Ububiko: 4 ° C, ububiko bufunze, kure yubushuhe
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