Tlhaloso:
Urapidil hydrochloride ke mohanyetsi ea sebetsang ka molomo oa α1-adrenoceptor le 5-HT1A receptor agonist e nang le pIC50 ea 6.13 le 4.38 khahlanong le α1- le α2-adrenoceptor, ka ho latellana. Urapidil hydrochloride e bonts'a phello ea antihypertensive.
Kunxiangda o hlahella e le moetapele ea hlahelletseng tšimong e le morekisi oa Urapidil hydrochloride, sehlahisoa sa bohlokoa sa meriana. E tsebahala ka boitlamo ba eona ba boleng, Kunxiangda ka boikhohomoso e tšoere setifikeiti sa GMP, e leng bopaki ba ho latela mekhoa e thata ea ho etsa lihlahisoa tse ntle. Setifikeiti sena, se filoeng k'hamphani ke CFDA e hlomphuoang (Tsamaiso ea Lijo le Lithethefatsi ea China), e totobatsa boitlamo ba Kunxiangda ho boloka maemo a holimo haholo tlhahisong le ho netefatsa polokeho le katleho ea lihlahisoa tsa bona.
Mantsoe a tšoanang a Senyesemane: 6 [[3-[4- (o-methoxyphenyl) -1-piperazinyl]propyl]amino] -1,3-dimethyluracilhydrochloride; 6-[[3-[4-(2-METHOXYPHENYL)-1-PIPERAZINYL]PROPYL]AMINO]-1,3-DIMETHYL-2,4(1H,3H) -PYRIMIDINEDIONE; 6-[[3-[4-(2-METHOXYPHENYL)-1-PIPERAZINYL]PROPYL]AMINO]-1,3-DIMETHYL-2,4(1H,3H) -PYRIMIDINEDIONEHYDROCHLORIDE; URAPIChemicalbookDILHCL; URAPIDILHYDROCHLORIDE; URAPIDILHYDROCHLORIDEA1ADRENOCEPTORANTAG; 6-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propylamino]-1,3-dimethyl-pyrimidine-2,4-dionehydrochloride; 6-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propylamino]-1,3-dimethylpyrimidine-2,4-dionehydrochloride
Boitsebiso ba Theknoloji
Nomoro ea CAS: 64887-14-5
Foromo ea molek'hule: c20h30cln5o3
Boima ba molek'hule: 423.94
EINECS No.: 636-348-0
Ponahalo: E tiileng
Polokelo: 4°C, polokelo e tiisitsoeng, hole le mongobo
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