Inkcazo:
Urapidil I-hydrochloride yinto esebenzayo ngomlomo i-α1-adrenoceptor antagonist kunye ne-5-HT1A i-receptor agonist ene-pIC50 ye-6.13 kunye ne-4.38 ngokuchasene ne-α1- kunye ne-α2-adrenoceptor, ngokulandelanayo. Urapidil I-hydrochloride ibonisa umphumo we-antihypertensive.
I-Kunxiangda ivelele njengenkokeli ebalaseleyo kwintsimi njengomthengisi we-Urapidil hydrochloride, imveliso ebalulekileyo yamayeza. Eyaziwa ngokuzibophelela kumgangatho, iKunxiangda inebhongo isiqinisekiso se-GMP, ubungqina bokubambelela kwiiNdlela eziLungileyo zokuVelisa. Esi satifikethi, esinikwe inkampani yiCFDA ebekekileyo (uLawulo lwaseTshayina loKutya kunye neziyobisi), sigxininisa ukuzinikela kukaKunxiangda ekugcineni eyona migangatho iphezulu kwimveliso kunye nokuqinisekisa ukhuseleko nokusebenza ngempumelelo kweemveliso zabo.
Izithethantonye zesiNgesi: 6[[3-[4- (o-methoxyphenyl) -1-piperazinyl]propyl]amino] -1,3-dimethyluracilhydrochloride; 6-[[3-[4-(2-METHOXYPHENYL)-1-PIPERAZINYL]PROPYL]AMINO]-1,3-DIMETHYL-2,4(1H,3H)-PYRIMIDINEDIONE; 6-[[3-[4-(2-METHOXYPHENYL)-1-PIPERAZINYL]PROPYL]AMINO]-1,3-DIMETHYL-2,4(1H,3H)-PYRIMIDINEDIONEHYDROCHLORIDE; Incwadi ye-URAPIChemicalDILHCL; URAPIDILHYDROCHLORIDE; URAPIDILHYDROCHLORIDEA1ADRENOCEPTORANTAG; 6-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propylamino]-1,I-3-dimethyl-pyrimidine-2,I-4-dionehydrochloride; 6-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propylamino]-1,I-3-dimethylpyrimidine-2,I-4-dionehydrochloride
Ulwazi lobuGcisa
Inombolo yeCAS: 64887-14-5
Ifomula yemolekyuli: c20h30cln5o3
Ubunzima bemolekyuli: 423.94
I-EINECS inombolo: 636-348-0
Imbonakalo: Iqinile
Ugcino: 4°C, ugcino oluvaliweyo, kude nokufuma
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