Bayani
Olprinone shine zaɓi na phosphodiesterase 3 (PDE3) mai hanawa. Ana amfani da Olprinone azaman wakili na cardiotonic tare da ingantaccen tasirin inotropic da vasodilating. An ba da rahoton Olprinone don inganta microcirculation da rage kumburi. Ana amfani da Olprinone sau da yawa don ƙara yawan fitarwa na zuciya bayan wucewar zuciya na zuciya (CPB). An shigar da Olprinone a cikin adadin 0.2 μg/kg/min lokacin da aka fara yaye daga CPB. Har ila yau, Olprinone ya nuna tasirin antioxidative da anti-mai kumburi a cikin meconium-induced oxidative huhu rauni.
Bayanin Fasaha:
Ma’ana: Olprinonehydrochloride-Loprinonehydrochloride; 3-pyridinecarbonitrile,1,2-dihydro-5-(imidazo(1,2-a) pyridin-6-yl)-6-methyl-2-o;e1020; xo-,monohydrochloride, monohydrate; OLPRINONEHCL;
Takaddun shaida: Takaddun shaida na GMP, CFDA
Tsarin kwayoyin halitta: C14H10N4O • HCl
Nauyin Formula: 286.7
Tsafta: ≥98%
Ƙirƙiri (Nemi canjin tsari)
SMILES na Canonical: CC1=C(C=C(C(=O)N1)C#N)C2=CN3C=CN=C3C=C2.Cl
Bayanin Ajiyewa & Ajiyewa:
Adana: -20°C
Aiki: Zazzabin ɗaki a nahiyar Amurka; na iya bambanta a wani wuri
Kwanciyar hankali: ≥ 4 shekaru
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