Katrangan
Olprinone minangka inhibitor selektif fosfodiesterase 3 (PDE3). Olprinone digunakake minangka agen kardiotonik kanthi efek inotropik lan vasodilating positif. Olprinone wis kacarita kanggo nambah microcirculation lan attenuate inflammation. Olprinone asring digunakake kanggo nambah output jantung sawise cardiopulmonary bypass (CPB). Olprinone diinfusake kanthi laju 0,2 μg/kg/menit nalika disapih saka CPB diwiwiti. Olprinone uga nuduhake efek antioksidatif lan anti-inflamasi sing kuat ing cedera paru-paru oksidatif meconium.
Informasi Teknis:
sinonim: Olprinonehydrochloride-Loprinonehydrochloride;3-pyridinecarbonitrile,1,2-dihidro-5-(imidazo(1,2-a) piridin-6-yl)-6-metil-2-o;e1020;xo-,monohidroklorida,monohidrat;OLPRINONEHCL;
Sertifikat: sertifikat GMP, CFDA
Formula Molekul: C14H10N4O • HCl
Bobot Formula: 286,7
Kemurnian: ≥98%
Formulasi (Request formulation change)
SENYUMAN kanonik: CC1=C(C=C(C(=O)N1)C#N)C2=CN3C=CN=C3C=C2.Cl
Informasi Pangiriman & Panyimpenan:
Panyimpenan: -20°C
Pengiriman: Suhu Kamar ing kontinental AS; bisa beda-beda ing papan liya
Stabilitas: ≥ 4 taun
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