Kufotokozera
Olprinone ndi choletsa cha phosphodiesterase 3 (PDE3) chosankha. Olprinone amagwiritsidwa ntchito ngati cardiotonic wothandizira wokhala ndi inotropic komanso vasodilating zotsatira. Olprinone yanenedwa kuti imathandizira microcirculation ndikuchepetsa kutupa. Olprinone nthawi zambiri amagwiritsidwa ntchito kuonjezera kutulutsa kwa mtima pambuyo pa cardiopulmonary bypass (CPB). Olprinone adalowetsedwa pamlingo wa 0.2 μg/kg/min pamene kuyamwa kuchokera ku CPB kunayambika. Olprinone yawonetsanso zotsatira zamphamvu za antioxidative ndi zotsutsana ndi zotupa mu meconium-induced oxidative mapapu kuvulala.
Zambiri Zaukadaulo:
Mawu ofanana ndi mawu: Olprinonehydrochloride-Loprinonehydrochloride;3-pyridinecarbonitrile,1,2-dihydro-5-(imidazo(1,2-a)pyridin-6-yl)-6-methyl-2-o;e1020;xo-,monohydrochloride,monohydrate;OLPRINONEHCL;
Certificate: Satifiketi ya GMP, CFDA
Molecular formula: C14H10N4O • HCl
Kulemera kwa formula: 286.7
Kuyera: ≥98%
Kupanga (Pemphani kusintha kwa mawonekedwe)
AKUmwetulira Ovomerezeka: CC1=C(C=C(C(=O)N1)C#N)C2=CN3C=CN=C3C=C2.Cl
Zotumiza ndi Kusunga:
Kusungirako: -20°C
Kutumiza: Kutentha kwa Zipinda mu continental US; zikhoza kusiyana kwina
Kukhazikika: ≥ 4 zaka
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