Deskripsyon
Olprinone se yon fosfodiesteraz selektif 3 (PDE3) inhibiteur. Olprinone yo itilize kòm ajan kadyotonik ak efè pozitif inotropik ak vazodilating. Olprinone yo te rapòte amelyore mikrosirkulasyon ak diminye enflamasyon. Olprinone souvan itilize pou ogmante pwodiksyon kadyak apre kontoune kadyopulmonè (CPB). Olprinone te enfuze nan yon pousantaj de 0.2 μg / kg / min lè sevraj soti nan CPB te kòmanse. Olprinone te montre tou pisan efè antioksidatif ak anti-enflamatwa nan aksidan nan poumon oksidatif mekonium-induit.
Enfòmasyon teknik:
Sinonim: Olprinonehydrochloride-Loprinonehydrochloride; 3-pyridinecarbonitrile,1,2-dihydro-5-(imidazo(1,2-a)piridin-6-yl)-6-methyl-2-o;e1020;xo-,monokloridrat,monoidrat;OLPRINONEHCL;
Sètifika: GMP sètifika, CFDA
Fòmil molekilè: C14H10N4O • HCl
Pwa fòmil: 286.7
Pite: ≥98%
Fòmasyon (Demann chanjman fòmilasyon)
SORI Kanonik: CC1=C(C=C(C(=O)N1)C#N)C2=CN3C=CN=C3C=C2.Cl
Enfòmasyon sou livrezon ak depo:
Depo: -20 ° C
Shipping: Tanperati chanm nan kontinantal Etazini; ka varye yon lòt kote
Estabilite: ≥ 4 ane
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