Fa'amatalaga
Olprinone o se phosphodiesterase filifilia 3 (PDE3) inhibitor. Olprinone o loʻo faʻaaogaina e fai ma sui o le cardiotonic ma lelei inotropic ma vasodilating aafiaga. Olprinone ua lipotia mai e faʻaleleia le microcirculation ma faʻaitiitia ai le mumū. Olprinone e masani ona faʻaaogaina e faʻateleina ai le gaosiga o le fatu pe a uma le cardiopulmonary bypass (CPB). Olprinone na faʻapipiʻiina i le fua o le 0.2 μg / kg / min pe a amata le susu mai le CPB. Olprinone ua faʻaalia foi le malosi o le antioxidative ma le anti-inflammatory aafiaga i le meconium-induced oxidative lung manua.
Fa'amatalaga Fa'atekinisi:
upu uiga tutusa: Olprinonehydrochloride-Loprinonehydrochloride;3-pyridinecarbonitrile,1,2-dihydro-5-(imidazo(1,2-a) piridin-6-yl) -6-methyl-2-o;e1020;xo-,monohydrochloride,monohydrate;OLPRINONEHCL;
Tusi Faamaonia: tusi faamaonia GMP, CFDA
Fuafuaga mole: C14H10N4O • HCl
Fuafuaga mamafa :286.7
Mama:≥98%
Fa'atulagaina(Talosaga suiga fa'atulagaina)
'ATA'ITA'I: CC1=C(C=C(C(=O)N1)C#N)C2=CN3C=CN=C3C=C2.Cl
Va'a & Teuina Fa'amatalaga:
Teuina: -20°C
Va'a: Temperature Room in continental US; e mafai ona eseese i se isi mea
Maumau: ≥ 4 tausaga
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