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bulk pharmaceutical intermediates

Olprinone Hydrochloride

Olprinone Hydrochloride
Description Olprinone is a selectiv

Nkọwa ngwaahịa

Mkpado ngwaahịa

Nkọwa

Olrinone bụ onye na-egbochi phosphodiesterase 3 (PDE3). A na-eji Olprinone dị ka onye na-ahụ maka cardiotonic nwere mmetụta inotropic na vasodilating dị mma. A kọwo Olprinone iji meziwanye microcirculation ma belata mbufụt. A na-ejikarị Olprinone na-amụba mmepụta obi mgbe ọ gafechara obi (CPB). A na-etinye Olprinone na ọnụego 0.2 μg / kg / min mgbe a malitere ịhapụ CPB. Olprinone egosikwala mmetụta antioxidative na mgbochi mkpali dị na meconium na-ebute mmerụ ahụ oxidative.

Ozi nka na ụzụ:

Ụdị okwu: Olprinonehydrochloride-Loprinonehydrochloride; 3-pyridinecarbonitrile,1,2-dihydro-5-(imidazo(1,2-a) pyridin-6-yl)-6-methyl-2-o;e1020; xo-,monohydrochloride,monohydrate;OLPRINONEHCL;

Asambodo: Asambodo GMP, CFDA

Ụdị molekụla: C14H10N4O • HCl

Ụdị arọ: 286.7

Ịdị ọcha: ≥98%

Nhazi(Chọọ mgbanwe nhazi usoro)

Ịchị ọchị: CC1=C(C=C(C(=O)N1)C#N)C2=CN3C=CN=C3C=C2.Cl

Ozi Mbupu & Nchekwa:

Nchekwa: -20C

Mbupu: Okpomọkụ ụlọ na kọntinent US; nwere ike ịdị iche n'ebe ọzọ

Nkwụsi ike: ≥ 4 afọ

 

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