Nkọwa
Olrinone bụ onye na-egbochi phosphodiesterase 3 (PDE3). A na-eji Olprinone dị ka onye na-ahụ maka cardiotonic nwere mmetụta inotropic na vasodilating dị mma. A kọwo Olprinone iji meziwanye microcirculation ma belata mbufụt. A na-ejikarị Olprinone na-amụba mmepụta obi mgbe ọ gafechara obi (CPB). A na-etinye Olprinone na ọnụego 0.2 μg / kg / min mgbe a malitere ịhapụ CPB. Olprinone egosikwala mmetụta antioxidative na mgbochi mkpali dị na meconium na-ebute mmerụ ahụ oxidative.
Ozi nka na ụzụ:
Ụdị okwu: Olprinonehydrochloride-Loprinonehydrochloride; 3-pyridinecarbonitrile,1,2-dihydro-5-(imidazo(1,2-a) pyridin-6-yl)-6-methyl-2-o;e1020; xo-,monohydrochloride,monohydrate;OLPRINONEHCL;
Asambodo: Asambodo GMP, CFDA
Ụdị molekụla: C14H10N4O • HCl
Ụdị arọ: 286.7
Ịdị ọcha: ≥98%
Nhazi(Chọọ mgbanwe nhazi usoro)
Ịchị ọchị: CC1=C(C=C(C(=O)N1)C#N)C2=CN3C=CN=C3C=C2.Cl
Ozi Mbupu & Nchekwa:
Nchekwa: -20C
Mbupu: Okpomọkụ ụlọ na kọntinent US; nwere ike ịdị iche n'ebe ọzọ
Nkwụsi ike: ≥ 4 afọ
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