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ʻO Olprinone kahi mea hoʻopaneʻe koho phosphodiesterase 3 (PDE3). Hoʻohana ʻia ʻo Olprinone e like me ka cardiotonic agent me ka inotropic maikaʻi a me nā hopena vasodilating. Ua hōʻike ʻia ʻo Olprinone e hoʻomaikaʻi i ka microcirculation a hoʻemi i ka mumū. Hoʻohana pinepine ʻia ʻo Olprinone e hoʻonui i ka puka o ka naʻau ma hope o ka cardiopulmonary bypass (CPB). Ua hoʻokomoʻiaʻo Olprinone ma kahi o 0.2 μg / kg / min i ka wā i hoʻomaka ai ka weaning mai CPB. Ua hōʻike pū ʻo Olprinone i nā hopena antioxidative a me nā hopena anti-inflammatory i ka meconium-induced lung lung lung.
ʻIkepili ʻenehana:
Nā huaʻōlelo like: Olprinonehydrochloride-Loprinonehydrochloride;3-pyridinecarbonitrile,1,2-dihydro-5-(imidazo(1,2-a)pyridin-6-yl)-6-methyl-2-o;e1020;xo-,monohydrochloride,monohydrate;OLPRINONEHCL;
Palapala: palapala GMP, CFDA
ʻAno Molekala: C14H10N4O • HCl
Kaumaha Kumu:286.7
Maʻemaʻe: ≥98%
Hoʻoponopono (Noi i ka hoʻololi hoʻololi)
ʻĀʻO KAONIKA: CC1=C(C=C(C(=O)N1)C#N)C2=CN3C=CN=C3C=C2.Cl
Hoʻouna a mālama ʻike:
Waihona: -20°C
Hoʻouna: lumi wela ma ka ʻāina ʻAmelika; hiki ke ʻokoʻa ma nā wahi ʻē aʻe
Paʻa: ≥ 4 makahiki
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