Ibisobanuro
Olprinone ni inhibitori ya fosifisiyose 3 (PDE3). Olprinone ikoreshwa nkumutima wumutima hamwe ningaruka nziza za inotropic na vasodilating. Olprinone yavuzwe ko izamura microcirculation kandi igabanya ubukana. Olprinone ikoreshwa kenshi mukongera umutima nyuma yumutima (CPB). Olprinone yashizwemo ku gipimo cya 0.2 μg / kg / min igihe konsa muri CPB byatangiraga. Olprinone yerekanye kandi ingaruka zikomeye za antioxydeid na anti-inflammatory mu gukomeretsa kwa meconium iterwa na okiside.
Amakuru ya tekiniki:
Synonyme: Olprinonehydrochloride-Loprinonehydrochloride; 3-pyridinecarbonitrile,1,2-dihydro-5- (imidazo (1),2-a) pyridin-6-yl) -6-methyl-2-o; e1020; xo-,monohydrochloride, monohydrate; OLPRINONEHCL;
Icyemezo: Icyemezo cya GMP, CFDA
Inzira ya molekulari: C.14H10N4O • HCl
Uburemere bwa formula: 286.7
Isuku: ≥98%
Gutegura (Gusaba guhindura formulaire)
Urwenya rwa Canonical: CC1 = C (C = C (C (= O) N1) C # N) C2 = CN3C = CN = C3C = C2.Cl
Kohereza & Ububiko Amakuru:
Ububiko: -20 ° C.
Kohereza: Ubushyuhe bwicyumba kumugabane wa Amerika; Birashobora gutandukana ahandi
Guhagarara: years imyaka 4
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